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2,4-Dichloropyrimidine in Pazopanib Intermediates: A Crucial Compound in Oncology API Synthesis

In modern pharmaceutical manufacturing, the development of complex APIs (Active Pharmaceutical Ingredients) demands high-purity and reliable chemical intermediates. One such essential compound is 2,4-Dichloropyrimidine, which plays a pivotal role in the synthesis of Pazopanib, a widely used anti-cancer drug.

Understanding 2,4-Dichloropyrimidine

2,4-Dichloropyrimidine is a pyrimidine derivative with the molecular formula C4H2Cl2N2. It features two chlorine atoms positioned at the 2nd and 4th carbon atoms of the pyrimidine ring, making it a versatile intermediate in pharmaceutical and agrochemical synthesis.

Due to its reactive nature and structural compatibility, this compound is commonly used in the development of kinase inhibitors, particularly Pazopanib, which is approved for treating renal cell carcinoma and soft tissue sarcoma.

Role in Pazopanib Synthesis

Pazopanib is a tyrosine kinase inhibitor that targets vascular endothelial growth factor receptors (VEGFRs), platelet-derived growth factor receptors (PDGFRs), and c-Kit, helping to block tumor angiogenesis. The synthesis process of Pazopanib involves multiple steps, with 2,4-Dichloropyrimidine being a key intermediate in constructing the drug’s core structure.

Using this intermediate helps ensure:

Enhanced chemical stability

Better reaction yield

High purity of the final API

Compatibility with large-scale production

Vidgastech – Reliable Supplier of Pharmaceutical Intermediates

Vidgastech is a leading manufacturer and global supplier of pharmaceutical intermediates, including 2,4-Dichloropyrimidine. We provide consistent quality, batch-to-batch purity, and scalable solutions for pharmaceutical R&D and production.

Our key strengths include:

✅ GMP-compliant production facilities
✅ Strict quality assurance processes
✅ Competitive pricing for bulk quantities
✅ On-time delivery worldwide
✅ Complete regulatory and technical documentation

Applications Beyond Pazopanib

While Pazopanib is a primary application, 2,4-Dichloropyrimidine is also used in:

Other kinase inhibitors

Antiviral and anti-inflammatory compounds

Research in pyrimidine-based drug discovery

Fine chemicals and specialty intermediates

Conclusion

In the landscape of oncology drug development, 2,4-Dichloropyrimidine continues to be a foundational compound, enabling the synthesis of powerful therapies like Pazopanib. As pharmaceutical research advances, the demand for high-quality intermediates grows—making Vidgastech a trusted partner for companies around the world.

🔗 To learn more or request a quote, visit:
👉 www.vidgastech.com

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